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Increased sensitivity to gemcitabine of P-glycoprotein and multidrug resistance-associated protein-overexpressing human cancer cell lines

Gemcitabine (2′,2′-difluorodeoxycytidine) is a deoxycytidine analogue that is activated by deoxycytidine kinase (dCK) to its monophosphate and subsequently to its triphosphate dFdCTP, which is incorporated into both RNA and DNA, leading to DNA damage. Multidrug resistance (MDR) is characterised by a...

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Dettagli Bibliografici
Autori principali: Bergman, A M, Pinedo, H M, Talianidis, I, Veerman, G, Loves, W J P, van der Wilt, C L, Peters, G J
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2003
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2741118/
https://ncbi.nlm.nih.gov/pubmed/12799644
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjc.6601011
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