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Increased sensitivity to gemcitabine of P-glycoprotein and multidrug resistance-associated protein-overexpressing human cancer cell lines

Gemcitabine (2′,2′-difluorodeoxycytidine) is a deoxycytidine analogue that is activated by deoxycytidine kinase (dCK) to its monophosphate and subsequently to its triphosphate dFdCTP, which is incorporated into both RNA and DNA, leading to DNA damage. Multidrug resistance (MDR) is characterised by a...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Bergman, A M, Pinedo, H M, Talianidis, I, Veerman, G, Loves, W J P, van der Wilt, C L, Peters, G J
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Nature Publishing Group 2003
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2741118/
https://ncbi.nlm.nih.gov/pubmed/12799644
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjc.6601011
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