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Molecular and physiologic basis of quinoline drug resistance in Plasmodium falciparum malaria

30 years before the discovery of the pfcrt gene, altered cellular drug accumulation in drug-resistant malarial parasites had been well documented. Heme released from catabolized hemoglobin was thought to be a key target for quinoline drugs, and additional modifications to quinoline drug structure in...

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Autor principal: Roepe, Paul D
Format: Artigo
Idioma:Inglês
Publicat: Future Medicine Ltd 2009
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2724744/
https://ncbi.nlm.nih.gov/pubmed/19416013
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2217/fmb.09.15
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