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Discovery of drug-resistant and drug-sensitizing mutations in the oncogenic PI3K isoform p110α

p110α (PIK3CA) is the most frequently mutated kinase in human cancer, and numerous drugs targeting this kinase are currently in pre-clinical development or early stage clinical trials. Clinical resistance to protein kinase inhibitors frequently results from point mutations that block drug binding; s...

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Bibliografske podrobnosti
Main Authors: Zunder, Eli R., Knight, Zachary A., Houseman, Benjamin T., Apsel, Beth, Shokat, Kevan M.
Format: Artigo
Jezik:Inglês
Izdano: 2008
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2720137/
https://ncbi.nlm.nih.gov/pubmed/18691552
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ccr.2008.06.014
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