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Drug Pressure Selected Mutations in HIV-1 Protease alter Flap Conformations

The flap conformations of two drug resistant HIV-1 protease constructs were characterized by molecular dynamic (MD) simulations and distance measurements with pulsed electron paramagnetic resonance (EPR) spectroscopy. MD simulations accurately regenerate the experimentally determined distance profil...

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Detalhes bibliográficos
Main Authors: Galiano, Luis, Ding, Fangyu, Veloro, Angelo M., Blackburn, Mandy E., Simmerling, Carlos, Fanucci, Gail E.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2705922/
https://ncbi.nlm.nih.gov/pubmed/19140783
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja807531v
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