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Replacement of a Thiourea-S with an Amidine-NH Donor Group in a Platinum–Acridine Antitumor Compound Reduces the Metal's Reactivity with Cysteine Sulfur

The reactivity of two DNA-targeted platinum–acridine conjugates with cysteine sulfur was studied. The conjugate containing an amidine-NH donor group cis to the chloride leaving group showed considerably reduced reactivity with N-acetylcysteine compared to the prototypical derivative containing a thi...

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Bibliografiske detaljer
Main Authors: Ma, Zhidong, Rao, Lu, Bierbach, Ulrich
Format: Artigo
Sprog:Inglês
Udgivet: 2009
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2693338/
https://ncbi.nlm.nih.gov/pubmed/19397321
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm900451y
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