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Molecular bases for the recognition of short peptide substrates and cysteine-directed modifications of human insulin-degrading enzyme

Insulin degrading enzyme (IDE) utilizes a large catalytic chamber to selectively bind and degrade peptide substrates such as insulin and amyloid β (Aβ). Tight interactions with substrates occur at an exosite located ~30Å away from the catalytic center that anchors the N-terminus of substrates to fac...

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Détails bibliographiques
Auteurs principaux: Malito, Enrico, Ralat, Luis A., Manolopoulou, Marika, Tsay, Julie L., Wadlington, Natasha L., Tang, Wei-Jen
Format: Artigo
Langue:Inglês
Publié: 2008
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2652632/
https://ncbi.nlm.nih.gov/pubmed/18986166
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi801192h
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