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Tyrosine sulfate isosteres of CCR5 N-terminus as tools for studying HIV-1 entry

The HIV-1 coreceptor CCR5 possesses tyrosine sulfate (TYS) residues at its N-terminus (Nt) that are required for binding HIV-1 gp120 and mediating viral entry. Using a 14-residue fragment of CCR5 Nt containing two TYS residues, we recently showed that CCR5 Nt binds gp120 through a conserved region s...

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Detalhes bibliográficos
Main Authors: Lam, Son N., Acharya, Priyamvada, Huang, Chih-Chin, Wyatt, Richard T., Kwong, Peter D., Bewley, Carole A.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2650494/
https://ncbi.nlm.nih.gov/pubmed/18952441
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2008.10.005
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