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The Design, Synthesis and Evaluation of Coumarin Ring Derivatives of the Novobiocin Scaffold that Exhibit Anti-proliferative Activity

[Image: see text] Novobiocin, a known DNA gyrase inhibitor, binds to a nucleotide-binding site located on the C-terminus of Hsp90 and induces degradation of Hsp90-dependent client proteins at ~700 μM in breast cancer cells (SkBr3). Although many analogues of novobiocin have been synthesized, it was...

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Detalhes bibliográficos
Main Authors: Donnelly, Alison C., Mays, Jared R., Burlison, Joseph A., Nelson, John T., Vielhauer, George, Holzbeierlein, Jeffrey, Blagg, Brian S. J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2646372/
https://ncbi.nlm.nih.gov/pubmed/18939877
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jo801312r
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