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Activation of G Protein–Coupled Receptors: Beyond Two-State Models and Tertiary Conformational Changes

Transformation of G protein–coupled receptors (GPCRs) from a quiescent to an active state initiates signal transduction. All GPCRs share a common architecture comprising seven transmembrane-spanning α-helices, which accommodates signal propagation from a diverse repertoire of external stimuli across...

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Detalhes bibliográficos
Main Authors: Park, Paul S.-H., Lodowski, David T., Palczewski, Krzysztof
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2639654/
https://ncbi.nlm.nih.gov/pubmed/17848137
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1146/annurev.pharmtox.48.113006.094630
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