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Activity of Indenoisoquinolines against African Trypanosomes

African trypanosomiasis (sleeping sickness), caused by protozoan Trypanosoma brucei species, is a debilitating disease that is lethal if untreated. Available drugs are antiquated, toxic, and compromised by emerging resistance. The indenoisoquinolines are a class of noncamptothecin topoisomerase IB p...

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Podrobná bibliografie
Hlavní autoři: Bakshi, Rahul P., Sang, Dongpei, Morrell, Andrew, Cushman, Mark, Shapiro, Theresa A.
Médium: Artigo
Jazyk:Inglês
Vydáno: American Society for Microbiology (ASM) 2009
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2612167/
https://ncbi.nlm.nih.gov/pubmed/18824603
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00650-07
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