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Structure of the ligand-binding domain of rat VDR in complex with the nonsecosteroidal vitamin D(3) analogue YR301

Vitamin D receptor (VDR) is a ligand-inducible hormone receptor that mediates 1α,25(OH)(2)D(3) action, regulating calcium and phosphate metabolism, induces potent cell differentiation activity and has immunosuppressive effects. Analogues of 1α,25(OH)(2)D(3) have been used clinically for some years....

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Autors principals: Kakuda, Shinji, Okada, Kazuhisa, Eguchi, Hiroshi, Takenouchi, Kazuya, Hakamata, Wataru, Kurihara, Masaaki, Takimoto-Kamimura, Midori
Format: Artigo
Idioma:Inglês
Publicat: International Union of Crystallography 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2581693/
https://ncbi.nlm.nih.gov/pubmed/18997319
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1107/S1744309108026754
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