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Activation of tyrosine kinases by mutation of the gatekeeper threonine

Protein kinases targeted by small-molecule inhibitors develop resistance through mutation of the ‘gatekeeper’ threonine residue of the active site. Here we show that the gatekeeper mutation in the cellular forms of c-ABL, c-SRC, platelet-derived growth factor receptor-α and -β, and epidermal growth...

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Hlavní autoři: Azam, Mohammad, Seeliger, Markus A, Gray, Nathanael S, Kuriyan, John, Daley, George Q
Médium: Artigo
Jazyk:Inglês
Vydáno: 2008
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2575426/
https://ncbi.nlm.nih.gov/pubmed/18794843
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nsmb.1486
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