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Cyclic Oxonitriles: Stereodivergent Grignard Addition-Alkylations

Sequential carbonyl addition-conjugate addition of Grignard reagents to cyclic 5–7–membered oxoalkenenitriles efficiently generates cyclic magnesiated nitriles. Alkylations of these magnesiated nitriles exhibit diastereoselectivities that depend intimately on the size of the carbocyclic ring: 5-memb...

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Detalhes bibliográficos
Main Authors: Fleming, Fraser F., Wei, Guoqing, Zhang, Zhiyu, Steward, Omar W.
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2553676/
https://ncbi.nlm.nih.gov/pubmed/17567075
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jo070678y
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