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Clerocidin selectively modifies the gyrase-DNA gate to induce irreversible and reversible DNA damage

Clerocidin (CL), a microbial diterpenoid, reacts with DNA via its epoxide group and stimulates DNA cleavage by type II DNA topoisomerases. The molecular basis of CL action is poorly understood. We establish by genetic means that CL targets DNA gyrase in the Gram-positive bacterium Streptococcus pneu...

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Detalhes bibliográficos
Main Authors: Pan, Xiao Su, Dias, Miriam, Palumbo, Manlio, Fisher, L. Mark
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2553588/
https://ncbi.nlm.nih.gov/pubmed/18723572
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkn539
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