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Synthesis of classical, four-carbon bridged 5-substituted furo[2,3-d]pyrimidine and 6-substituted pyrrolo[2,3-d]pyrimidine analogues as antifolates1

We report, for the first time, the biological activities of four carbon atom bridged classical antifolates on dihydrofolate reductase (DHFR), thymidylate synthase (TS) and folylpolyglutamate synthetase (FPGS) as well as on antitumor activity. Extension of the bridge homologation studies of classical...

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Detalles Bibliográficos
Main Authors: Gangjee, Aleem, Zeng, Yibin, McGuire, John J., Kisliuk, Roy L.
Formato: Artigo
Idioma:Inglês
Publicado: 2005
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2538949/
https://ncbi.nlm.nih.gov/pubmed/16078850
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm058213s
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