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Substituted Pyrrolo[2,3-d]pyrimidines as Cryptosporidium hominis Thymidylate Synthase Inhibitors

Cryptosporidiosis, a gastrointestinal disease caused by a protozoan Cryptosporidium hominis is often fatal in immunocompromised individuals. There is little clinical data to show that the existing treatment by nitazoxanide and paromomycin is effective in immunocompromised individuals(1, 2). Thymidyl...

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Autori principali: Kumar, Vidya P., Frey, Kathleen M., Wang, Yiqiang, Jain, Hitesh K., Gangjee, Aleem, Anderson, Karen S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3853131/
https://ncbi.nlm.nih.gov/pubmed/23927969
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.07.037
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