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Oxonitriles: A Grignard Addition-Acylation Route to Enamides

Sequential addition of three different Grignard reagents and pivaloyl chloride to 3-oxo-1-cyclohexene-1-carbonitrile installs four new bonds to generate a diverse array of cyclic enamides. Remarkably, formation of the C-magnesiated nitrile intermediate is followed by preferential acylation by pivalo...

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Autori principali: Fleming, Fraser F., Wei, Guoqing, Zhang, Zhiyu, Steward, Omar W.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2006
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2518779/
https://ncbi.nlm.nih.gov/pubmed/17020332
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol0619765
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