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Kinase packing defects as drug targets
Protein packing defects constitute structural singularities arising from backbone overexposure to water. Such features may be targeted in kinase-inhibitor design to achieve specificity, to control cross reactivity and to overcome drug resistant mutations. Protein kinases constitute major targets in...
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| Main Authors: | , |
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| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
2007
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2136416/ https://ncbi.nlm.nih.gov/pubmed/17993409 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drudis.2007.09.009 |
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