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Crystal Structure of the Geobacillus stearothermophilus Carboxylesterase Est55 and Its Activation of Prodrug CPT-11

Several mammalian carboxylesterases were shown to activate the prodrug irinotecan (CPT-11) to produce SN-38, a topoisomerase inhibitor used in cancer therapy. However, the potential use of bacterial carboxylesterases, which have the advantage of high stability, has not been explored. We present the...

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Main Authors: Liu, Ping, Ewis, Hosam E., Tai, Phang C., Lu, Chung-Dar, Weber, Irene T.
格式: Artigo
語言:Inglês
出版: 2006
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC1950602/
https://ncbi.nlm.nih.gov/pubmed/17239398
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jmb.2006.12.067
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