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Different flecainide sensitivity of hNa(v)1.4 channels and myotonic mutants explained by state-dependent block

Flecainide, a class IC antiarrhythmic, was shown to improve myotonia caused by sodium channel mutations in situations where the class IB antiarrhythmic drug mexiletine was less efficient. Yet little is known about molecular interactions between flecainide and human skeletal muscle sodium (hNa(v)1.4)...

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Hlavní autoři: Desaphy, Jean-François, Luca, Annamaria D E, Didonna, Maria Paola, George, Alfred L, Camerino, Diana Conte
Médium: Artigo
Jazyk:Inglês
Vydáno: Blackwell Science Inc 2004
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1664778/
https://ncbi.nlm.nih.gov/pubmed/14608015
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1113/jphysiol.2003.046995
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