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Understanding tubulin–Taxol interactions: Mutations that impart Taxol binding to yeast tubulin

We have successfully used mutagenesis to engineer Taxol (paclitaxel) binding activity in Saccharomyces cerevisiae tubulin. Taxol, a successful antitumor agent, acts by promoting tubulin assembly and stabilizing microtubules. Several structurally diverse antimitotic compounds, including the epothilon...

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Библиографические подробности
Главные авторы: Gupta, Mohan L., Bode, Claudia J., Georg, Gunda I., Himes, Richard H.
Формат: Artigo
Язык:Inglês
Опубликовано: National Academy of Sciences 2003
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC164457/
https://ncbi.nlm.nih.gov/pubmed/12740436
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1131967100
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