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Transport and uptake of nateglinide in Caco-2 cells and its inhibitory effect on human monocarboxylate transporter MCT1

1. Nateglinide, a novel oral hypoglycemic agent, rapidly reaches the maximum serum concentration after oral administration, suggesting that it is rapidly absorbed in the gastrointestinal tract. The aim of this work is to clarify the intestinal absorption mechanism of nateglinide by means of in vitro...

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Autors principals: Okamura, Atsuko, Emoto, Akiko, Koyabu, Noriko, Ohtani, Hisakazu, Sawada, Yasufumi
Format: Artigo
Idioma:Inglês
Publicat: 2002
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573497/
https://ncbi.nlm.nih.gov/pubmed/12237260
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0704875
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