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Transport and uptake of nateglinide in Caco-2 cells and its inhibitory effect on human monocarboxylate transporter MCT1

1. Nateglinide, a novel oral hypoglycemic agent, rapidly reaches the maximum serum concentration after oral administration, suggesting that it is rapidly absorbed in the gastrointestinal tract. The aim of this work is to clarify the intestinal absorption mechanism of nateglinide by means of in vitro...

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Autori principali: Okamura, Atsuko, Emoto, Akiko, Koyabu, Noriko, Ohtani, Hisakazu, Sawada, Yasufumi
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2002
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573497/
https://ncbi.nlm.nih.gov/pubmed/12237260
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0704875
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