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Histamine H(3)-receptor-mediated [(35)S]GTPγ[S] binding: evidence for constitutive activity of the recombinant and native rat and human H(3) receptors

1. Constitutive activity of the recombinant and native rat and human H(3) receptors (H(3)Rs) was studied using H(3)R-mediated [(35)S]GTPγ[S] binding and [(3)H]-arachidonic acid release. 2. Ciproxifan, an inverse agonist at the rat H(3)R (rH(3)R), decreased [(3)H]arachidonic acid release from CHO cel...

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Bibliographic Details
Main Authors: Rouleau, A, Ligneau, X, Tardivel-Lacombe, J, Morisset, S, Gbahou, F, Schwartz, J -C, Arrang, J -M
Format: Artigo
Language:Inglês
Published: 2002
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573152/
https://ncbi.nlm.nih.gov/pubmed/11815373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0704490
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