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The nonpeptide B(2) receptor antagonist FR173657: inhibition of effects of bradykinin related to its role in nociception

1. The nonpeptide bradykinin B(2) receptor antagonist, FR173657 ((E)-3-(6-acetamido-3-pyridyl)-N-[N-(2, 4-dichloro-3-[(2-methyl-8-quinolinyl) oxymethyl] phenyl]-N-methylaminocarbonylmethyl] acrylamide), was tested in models involving bradykinin-induced activation of primary afferent neurones in vitr...

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Dettagli Bibliografici
Autori principali: Griesbacher, Thomas, Amann, Rainer, Sametz, Wolfgang, Diethart, Sabine, Juan, Heinz
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1998
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1565494/
https://ncbi.nlm.nih.gov/pubmed/9720808
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0701938
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