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Thiazolidinone CFTR inhibitor identified by high-throughput screening blocks cholera toxin–induced intestinal fluid secretion

Secretory diarrhea is the leading cause of infant death in developing countries and a major cause of morbidity in adults. The cystic fibrosis transmembrane conductance regulator (CFTR) protein is required for fluid secretion in the intestine and airways and, when defective, causes the lethal genetic...

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Autors principals: Ma, Tonghui, Thiagarajah, Jay R., Yang, Hong, Sonawane, Nitin D., Folli, Chiara, Galietta, Luis J.V., Verkman, A.S.
Format: Artigo
Idioma:Inglês
Publicat: American Society for Clinical Investigation 2002
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC151633/
https://ncbi.nlm.nih.gov/pubmed/12464670
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/JCI16112
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