Nalaganje...

THIAZOLIDINONE CFTR INHIBITORS WITH IMPROVED WATER SOLUBILITY IDENTIFIED BY STRUCTURE-ACTIVITY ANALYSIS

The thiazolidinone 3-[(3-trifluoromethyl)phenyl]-5-[(4-carboxyphenyl)methylene]-2-thioxo-4-thiazolidinone (CFTR(inh)-172) inhibits cystic fibrosis transmembrane conductance regulator (CFTR) chloride channel conductance with submicromolar affinity and blocks cholera toxin-induced intestinal fluid sec...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
Main Authors: Sonawane, N.D., Verkman, A.S.
Format: Artigo
Jezik:Inglês
Izdano: 2008
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2577561/
https://ncbi.nlm.nih.gov/pubmed/18691893
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2008.07.044
Oznake: Označite
Brez oznak, prvi označite!