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G Protein-coupled Receptor Kinase 2 Negatively Regulates Chemokine Signaling at a Level Downstream from G Protein Subunits

The G protein-coupled receptor kinase 2 (GRK2) phosphorylates and desensitizes ligand-activated G protein-coupled-receptors. Here, evidence is shown for a novel role of GRK2 in regulating chemokine-mediated signals. The presence of increased levels of GRK2 in human embryonic kidney (HEK) 293 cells p...

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Detalhes bibliográficos
Main Authors: Jiménez-Sainz, M. Carmen, Murga, Cristina, Kavelaars, Annemieke, Jurado-Pueyo, María, Krakstad, Beate F., Heijnen, Cobi J., Mayor, Federico, Aragay, Anna M.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Cell Biology 2006
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1345643/
https://ncbi.nlm.nih.gov/pubmed/16221891
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1091/mbc.E05-05-0399
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