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Probing cathepsin K activity with a selective substrate spanning its active site.

The limited availability of highly selective cathepsin substrates seriously impairs studies designed to monitor individual cathepsin activities in biological samples. Among mammalian cysteine proteases, cathepsin K has a unique preference for a proline residue at P2, the primary determinant of its s...

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Detaylı Bibliyografya
Asıl Yazarlar: Lecaille, Fabien, Weidauer, Enrico, Juliano, Maria A, Brömme, Dieter, Lalmanach, Gilles
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2003
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC1223680/
https://ncbi.nlm.nih.gov/pubmed/12837132
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20030468
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