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Lysine(164)alpha of protein farnesyltransferase is important for both CaaX substrate binding and catalysis.

Protein farnesyltransferase (FTase) catalyses the formation of a thioether linkage between proteins containing a C-terminal CaaX motif and a 15-carbon isoprenoid. The involvement of substrates such as oncogenic Ras proteins in tumour formation has led to intense efforts in targeting this enzyme for...

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Bibliografski detalji
Glavni autori: Hightower, K E, De, S, Weinbaum, C, Spence, R A, Casey, P J
Format: Artigo
Jezik:Inglês
Izdano: 2001
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC1222265/
https://ncbi.nlm.nih.gov/pubmed/11736652
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