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Pharmacological Properties of a New Antimalarial Bisthiazolium Salt, T3, and a Corresponding Prodrug, TE3

A new approach to malarial chemotherapy based on quaternary ammonium that targets membrane biogenesis during intraerythrocytic Plasmodium falciparum development has recently been developed. To increase the bioavailability, nonionic chemically modified prodrugs were synthesized. In this paper, the ph...

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Detalhes bibliográficos
Main Authors: Nicolas, Olivier, Margout, Delphine, Taudon, Nicolas, Wein, Sharon, Calas, Michèle, Vial, Henri J., Bressolle, Françoise M. M.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2005
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1195427/
https://ncbi.nlm.nih.gov/pubmed/16127032
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.49.9.3631-3639.2005
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