Aminopyrazole Carboxamide Bruton’s Tyrosine Kinase Inhibitors. Irreversible to Reversible Covalent Reactive Group Tuning

ανά Schnute, Mark E., Benoit, Stephen E., Buchler, Ingrid P., Caspers, Nicole, Grapperhaus, Margaret L., Han, Seungil, Hotchandani, Rajeev, Huang, Nelson, Hughes, Robert O., Juba, Brian M., Kim, Kyung-Hee, Liu, Erica, McCarthy, Erin, Messing, Dean, Miyashiro, Joy S., Mohan, Shashi, O’Connell, Thomas N., Ohren, Jeffrey F., Parikh, Mihir D., Schmidt, Michelle, Selness, Shaun R., Springer, John R., Thanabal, Venkataraman, Trujillo, John I., Walker, Daniel P., Wan, Zhao-Kui, Withka, Jane M., Wittwer, Arthur J., Wood, Nancy L., Xing, Li, Zapf, Christoph W., Douhan, John
Τόπος έκδοσης ACS Med Chem Lett (2018)

Discovery of an Oral Potent Selective Inhibitor of Hematopoietic Prostaglandin D Synthase (HPGDS)

ανά Carron, Chris P., Trujillo, John I., Olson, Kirk L., Huang, Wei, Hamper, Bruce C., Dice, Tom, Neal, Bradley E., Pelc, Matthew J., Day, Jacqueline E., Rohrer, Douglas C., Kiefer, James R., Moon, Joseph B., Schweitzer, Barbara A., Blake, Tanisha D., Turner, Steve R., Woerndle, Rhonda, Case, Brenda L., Bono, Christine P., Dilworth, Vickie M., Funckes-Shippy, Christie L., Hood, Becky L., Jerome, Gina M., Kornmeier, Christine M., Radabaugh, Melissa R., Williams, Melanie L., Davies, Michael S., Wegner, Craig D., Welsch, Dean J., Abraham, William M., Warren, Chad J., Dowty, Martin E., Hua, Fengmei, Zutshi, Anup, Yang, Jerry Z., Thorarensen, Atli
Έκδοση 2010