Study of Adrenocorticotropic Hormone Conformation by Evaluation of Intramolecular Resonance Energy Transfer in N(ε)-Dansyllysine(21)-ACTH-(1-24)-Tetrakosipeptide

Por Schiller, Peter W.
Publicado em 1972

Opioid peptide-derived analgesics

Por Schiller, Peter W.
Publicado em 2005

Bi- or multifunctional peptide drugs

Por Schiller, Peter W.
Publicado em 2009

Synthesis and Pharmacological Evaluation of Highly Potent [Dmt(1)]DALDA Analogs

Por Reddy, P. Anantha, Lewin, Anita H., Schiller, Peter W.
Publicado em 2009

Bifunctional μ/δ Opioid Peptides: Variation of the Type and Length of the Linker Connecting the Two Components

Por Ding, Jinguo, Lemieux, Carole, Chung, Nga N., Schiller, Peter W.
Publicado em 2012

Tolerance develops in spinal cord, but not in brain with chronic [Dmt(1)]DALDA treatment

Por Ben, Yong, Smith, Andrew P, Schiller, Peter W, Lee, Nancy M
Publicado em 2004

Histone Deacetylase-3 Activation Promotes Tumor Necrosis Factor-α (TNF-α) Expression in Cardiomyocytes during Lipopolysaccharide Stimulation

Por Zhu, Huaqing, Shan, Limei, Schiller, Peter W., Mai, Antonello, Peng, Tianqing
Publicado em 2010

Endocytic Profiles of δ-Opioid Receptor Ligands Determine the Duration of Rapid but Not Sustained cAMP Responses

Por Tudashki, Hanieh Bagheri, Robertson, Derek N., Schiller, Peter W., Pineyro, Graciela
Publicado em 2014

One-Pot Isomerization–Cross Metathesis–Reduction (ICMR) Synthesis of Lipophilic Tetrapeptides

Por Jida, Mouhamad, Betti, Cecilia, Schiller, Peter W., Tourwé, Dirk, Ballet, Steven
Publicado em 2014

Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists

Por Berezowska, Irena, Lemieux, Carole, Chung, Nga N., Ding, Jinguo, Schiller, Peter W.
Publicado em 2012

Superior analgesic effect of H-Dmt-D-Arg-Phe-Lys-NH(2) ([Dmt(1)]DALDA), a multifunctional opioid peptide, compared to morphine in a rat model of neuropathic pain

Por Shimoyama, Megumi, Schiller, Peter W., Shimoyama, Naohito, Toyama, Satoshi, Szeto, Hazel H.
Publicado em 2012

Dicarba Analogues of the Cyclic Enkephalin Peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) Retain High Opioid Activity

Por Berezowska, Irena, Chung, Nga N., Lemieux, Carole, Wilkes, Brian C., Schiller, Peter W.
Publicado em 2007

Stereoselective Synthesis of (3S)- and (3R)-3-Hydroxy-3-(2,6-Dimethyl-4-Hydroxyphenyl)Propanoic Acid and its Incorporation into a Cyclic Enkephalin Analogue

Por Weltrowska, Grazyna, Lemieux, Carole, Chung, Nga N., Wilkes, Brian C., Schiller, Peter W.
Publicado em 2009

Cyclic Opioid Peptide Agonists and Antagonists Obtained Via Ring-Closing Metathesis

Por Berezowska, Irena, Lemieux, Carole, Chung, Nga N., Wilkes, Brian C., Schiller, Peter W.
Publicado em 2009

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr(1)

Por Berezowska, Irena, Chung, Nga N., Lemieux, Carole, Wilkes, Brian C., Schiller, Peter W.
Publicado em 2009

Molecular Pharmacology of δ-Opioid Receptors

Por Gendron, Louis, Cahill, Catherine M., von Zastrow, Mark, Schiller, Peter W., Pineyro, Graciela
Publicado no Pharmacol Rev (2016)

Conformation-activity relationships of cyclo-constrained μ/δ opioid agonists derived from the N-terminal tetrapeptide segment of dermorphin/deltorphin

Por Ciarkowski, Jerzy, Czaplewski, Cezary, Łuczak, Sylwia, Rodziewicz-Motowidło, Sylwia, Berezowska, Irena, Schiller, Peter W.
Publicado em 2009

N-Methylated Cyclic Enkephalin Analogues Retain High Opioid Receptor Binding Affinity

Por Weltrowska, Grazyna, Berezowska, Irena, Lemieux, Carole, Chung, Nga N., Wilkes, Brian C., Schiller, Peter W.
Publicado em 2009

N-terminal guanidinylation of TIPP (Tyr-Tic-Phe-Phe) peptides results in major changes of the opioid activity profile

Por Weltrowska, Grazyna, Nguyen, Thi M.-D., Chung, Nga N., Wilkes, Brian C., Schiller, Peter W.
Publicado em 2013

Bioluminescence Resonance Energy Transfer Assays Reveal Ligand-specific Conformational Changes within Preformed Signaling Complexes Containing δ-Opioid Receptors and Heterotrimeric...

Por Audet, Nicolas, Galés, Céline, Archer-Lahlou, Élodie, Vallières, Marc, Schiller, Peter W., Bouvier, Michel, Pineyro, Graciela
Publicado em 2008