Design and Synthesis of Potent Macrocyclic HIV-1 Protease Inhibitors Involving P1-P2 Ligands

Por Ghosh, Arun K., Schiltz, Gary E., Rusere, Linah N., Osswald, Heather L., Walters, D. Eric, Amano, Masayuki, Mitsuya, Hiroaki
Publicado em 2014

Quinoxaline-Based Linear HCV NS3/4A Protease Inhibitors Exhibit Potent Activity against Drug Resistant Variants

Por Rusere, Linah N., Matthew, Ashley N., Lockbaum, Gordon J., Jahangir, Muhammad, Newton, Alicia, Petropoulos, Christos J., Huang, Wei, Kurt Yilmaz, Nese, Schiffer, Celia A., Ali, Akbar
Publicado no ACS Med Chem Lett (2018)

HIV-1 Protease Inhibitors Incorporating Stereochemically Defined P2′ Ligands to Optimize Hydrogen Bonding in the Substrate Envelope

Por Rusere, Linah N., Lockbaum, Gordon J., Lee, Sook-Kyung, Henes, Mina, Kosovrasti, Klajdi, Spielvogel, Ean, Nalivaika, Ellen A., Swanstrom, Ronald, Yilmaz, Nese Kurt, Schiffer, Celia A., Ali, Akbar
Publicado no J Med Chem (2019)

Structural Adaptation of Darunavir Analogs Against Primary Mutations in HIV-1 Protease

Por Lockbaum, Gordon J., Leidner, Florian, Rusere, Linah N., Henes, Mina, Kosovrasti, Klajdi, Nachum, Gily S., Nalivaika, Ellen A., Bolon, Daniel N.A., Ali, Akbar, Yilmaz, Nese Kurt, Schiffer, Celia A.
Publicado no ACS Infect Dis (2018)

Correction to Structural Adaptation of Darunavir Analogues against Primary Mutations in HIV-1 Protease.

Por Lockbaum, Gordon J., Leidner, Florian, Rusere, Linah N., Henes, Mina, Kosovrasti, Klajdi, Nachum, Gily S., Nalivaika, Ellen A., Bolon, Daniel N.A., Ali, Akbar, Yilmaz, Nese Kurt, Schiffer, Celia A.
Publicado no ACS Infect Dis (2019)