4-Hydroxypiperidines and Their Flexible 3-(Amino)propyloxy Analogues as Non-Imidazole Histamine H(3) Receptor Antagonist: Further Structure–Activity Relationship Exploration and In...

par Olszewska, Beata, Stasiak, Anna, McNaught Flores, Daniel, Fogel, Wiesława Agnieszka, Leurs, Rob, Walczyński, Krzysztof
Publié dans Int J Mol Sci (2018)

Non-Imidazole Histamine H(3) Ligands. Part VII. Synthesis, In Vitro and In Vivo Characterization of 5-Substituted-2-thiazol-4-n-propylpiperazines

par Guryn, Roman, Staszewski, Marek, Stasiak, Anna, McNaught Flores, Daniel, Fogel, Wiesława Agnieszka, Leurs, Rob, Walczyński, Krzysztof
Publié dans Molecules (2018)

Function-specific virtual screening for GPCR ligands using a combined scoring method

par Kooistra, Albert J., Vischer, Henry F., McNaught-Flores, Daniel, Leurs, Rob, de Esch, Iwan J. P., de Graaf, Chris
Publié dans Sci Rep (2016)

Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H(3) receptor antag...

par Staszewski, Marek, Stasiak, Anna, Karcz, Tadeusz, McNaught Flores, Daniel, Fogel, Wiesława Agnieszka, Kieć-Kononowicz, Katarzyna, Leurs, Rob, Walczyński, Krzysztof
Publié dans Medchemcomm (2019)