Allosteric modulation of G protein‐coupled receptors by amiloride and its derivatives. Perspectives for drug discovery?

由 Massink, Arnault, Amelia, Tasia, Karamychev, Alex, IJzerman, Adriaan P.
發表在 Med Res Rev (2019)

In search of novel ligands using a structure-based approach: a case study on the adenosine A(2A) receptor

由 Lenselink, Eelke B., Beuming, Thijs, van Veen, Corine, Massink, Arnault, Sherman, Woody, van Vlijmen, Herman W. T., IJzerman, Adriaan P.
發表在 J Comput Aided Mol Des (2016)

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A(1) adenosine receptor

由 Guo, Dong, Venhorst, Suzanne N, Massink, Arnault, van Veldhoven, Jacobus P D, Vauquelin, Georges, IJzerman, Adriaan P, Heitman, Laura H
發表在 Br J Pharmacol (2014)

Sodium Ion Binding Pocket Mutations and Adenosine A(2A) Receptor Function

由 Massink, Arnault, Gutiérrez-de-Terán, Hugo, Lenselink, Eelke B., Ortiz Zacarías, Natalia V., Xia, Lizi, Heitman, Laura H., Katritch, Vsevolod, Stevens, Raymond C., IJzerman, Adriaan P.
發表在 Mol Pharmacol (2015)

The role of a sodium ion binding site in the allosteric modulation of the A(2A) adenosine G protein-coupled receptor

由 Gutiérrez-de-Terán, Hugo, Massink, Arnault, Rodríguez, David, Liu, Wei, Han, Gye Won, Joseph, Jeremiah S., Katritch, Ilia, Heitman, Laura H., Xia, Lizi, IJzerman, Adriaan P., Cherezov, Vadim, Katritch, Vsevolod, Stevens, Raymond C.
出版 2013