Allosteric modulation of G protein‐coupled receptors by amiloride and its derivatives. Perspectives for drug discovery?

Bằng Massink, Arnault, Amelia, Tasia, Karamychev, Alex, IJzerman, Adriaan P.
Xuất bản năm Med Res Rev (2019)

In search of novel ligands using a structure-based approach: a case study on the adenosine A(2A) receptor

Bằng Lenselink, Eelke B., Beuming, Thijs, van Veen, Corine, Massink, Arnault, Sherman, Woody, van Vlijmen, Herman W. T., IJzerman, Adriaan P.
Xuất bản năm J Comput Aided Mol Des (2016)

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A(1) adenosine receptor

Bằng Guo, Dong, Venhorst, Suzanne N, Massink, Arnault, van Veldhoven, Jacobus P D, Vauquelin, Georges, IJzerman, Adriaan P, Heitman, Laura H
Xuất bản năm Br J Pharmacol (2014)

Sodium Ion Binding Pocket Mutations and Adenosine A(2A) Receptor Function

Bằng Massink, Arnault, Gutiérrez-de-Terán, Hugo, Lenselink, Eelke B., Ortiz Zacarías, Natalia V., Xia, Lizi, Heitman, Laura H., Katritch, Vsevolod, Stevens, Raymond C., IJzerman, Adriaan P.
Xuất bản năm Mol Pharmacol (2015)

The role of a sodium ion binding site in the allosteric modulation of the A(2A) adenosine G protein-coupled receptor

Bằng Gutiérrez-de-Terán, Hugo, Massink, Arnault, Rodríguez, David, Liu, Wei, Han, Gye Won, Joseph, Jeremiah S., Katritch, Ilia, Heitman, Laura H., Xia, Lizi, IJzerman, Adriaan P., Cherezov, Vadim, Katritch, Vsevolod, Stevens, Raymond C.
Được phát hành 2013