Allosteric modulation of G protein‐coupled receptors by amiloride and its derivatives. Perspectives for drug discovery?

द्वारा Massink, Arnault, Amelia, Tasia, Karamychev, Alex, IJzerman, Adriaan P.
में प्रकाशित Med Res Rev (2019)

In search of novel ligands using a structure-based approach: a case study on the adenosine A(2A) receptor

द्वारा Lenselink, Eelke B., Beuming, Thijs, van Veen, Corine, Massink, Arnault, Sherman, Woody, van Vlijmen, Herman W. T., IJzerman, Adriaan P.
में प्रकाशित J Comput Aided Mol Des (2016)

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A(1) adenosine receptor

द्वारा Guo, Dong, Venhorst, Suzanne N, Massink, Arnault, van Veldhoven, Jacobus P D, Vauquelin, Georges, IJzerman, Adriaan P, Heitman, Laura H
में प्रकाशित Br J Pharmacol (2014)

Sodium Ion Binding Pocket Mutations and Adenosine A(2A) Receptor Function

द्वारा Massink, Arnault, Gutiérrez-de-Terán, Hugo, Lenselink, Eelke B., Ortiz Zacarías, Natalia V., Xia, Lizi, Heitman, Laura H., Katritch, Vsevolod, Stevens, Raymond C., IJzerman, Adriaan P.
में प्रकाशित Mol Pharmacol (2015)

The role of a sodium ion binding site in the allosteric modulation of the A(2A) adenosine G protein-coupled receptor

द्वारा Gutiérrez-de-Terán, Hugo, Massink, Arnault, Rodríguez, David, Liu, Wei, Han, Gye Won, Joseph, Jeremiah S., Katritch, Ilia, Heitman, Laura H., Xia, Lizi, IJzerman, Adriaan P., Cherezov, Vadim, Katritch, Vsevolod, Stevens, Raymond C.
प्रकाशित 2013