Discovery of Tertiary Amine and Indole Derivatives as Potent RORγt Inverse Agonists

von Yang, Ting, Liu, Qian, Cheng, Yaobang, Cai, Wei, Ma, Yingli, Yang, Liuqing, Wu, Qianqian, Orband-Miller, Lisa A., Zhou, Ling, Xiang, Zhijun, Huxdorf, Melanie, Zhang, Wei, Zhang, Jing, Xiang, Jia-Ning, Leung, Stewart, Qiu, Yang, Zhong, Zhong, Elliott, John D., Lin, Xichen, Wang, Yonghui
Veröffentlicht 2013

Discovery of Biaryl Amides as Potent, Orally Bioavailable, and CNS Penetrant RORγt Inhibitors

von Wang, Yonghui, Cai, Wei, Cheng, Yaobang, Yang, Ting, Liu, Qian, Zhang, Guifeng, Meng, Qinghua, Han, Fangbin, Huang, Yafei, Zhou, Ling, Xiang, Zhijun, Zhao, Yong-Gang, Xu, Yan, Cheng, Ziqiang, Lu, Sijie, Wu, Qianqian, Xiang, Jia-Ning, Elliott, John D., Leung, Stewart, Ren, Feng, Lin, Xichen
Veröffentlicht in ACS Med Chem Lett (2015)