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Structural insights into JAK2 inhibition by ruxolitinib, fedratinib, and derivatives thereof

The discovery that aberrant activity of Janus kinase 2 (JAK2) is a driver of myeloproliferative neoplasms (MPNs) has led to significant efforts to develop small molecule inhibitors for this patient population. Ruxolitinib and fedratinib have been approved for use in MPN patients, while baricitinib,...

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Bibliografiske detaljer
Udgivet i:J Med Chem
Main Authors: Davis, Ryan R., Li, Baoli, Yun, Sang Y., Chan, Alice, Nareddy, Pradeep, Gunawan, Steven, Ayaz, Muhammad, Lawrence, Harshani R., Reuther, Gary W., Lawrence, Nicholas J., Schönbrunn, Ernst
Format: Artigo
Sprog:Inglês
Udgivet: 2021
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8327781/
https://ncbi.nlm.nih.gov/pubmed/33570945
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01952
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