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Purinergic Signaling: Impact of GPCR Structures on Rational Drug Design

The purinergic signaling system includes membrane-bound receptors for extracellular purines and pyrimidines, and enzymes/transporters that regulate receptor activation by endogenous agonists. Receptors include: adenosine (A(1), A(2A), A(2B) and A(3)) and P2Y (P2Y(1) P2Y(2), P2Y(4), P2Y(6), P2Y(11),...

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Détails bibliographiques
Publié dans:ChemMedChem
Auteurs principaux: Salmaso, Veronica, Jacobson, Kenneth A.
Format: Artigo
Langue:Inglês
Publié: 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC8276773/
https://ncbi.nlm.nih.gov/pubmed/32803849
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.202000465
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