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In Silico Drug Design for Purinergic GPCRs: Overview on Molecular Dynamics Applied to Adenosine and P2Y Receptors

Molecular modeling has contributed to drug discovery for purinergic GPCRs, including adenosine receptors (ARs) and P2Y receptors (P2YRs). Experimental structures and homology modeling have proven to be useful in understanding and predicting structure activity relationships (SAR) of agonists and anta...

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Dettagli Bibliografici
Pubblicato in:Biomolecules
Autori principali: Salmaso, Veronica, Jacobson, Kenneth A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7356333/
https://ncbi.nlm.nih.gov/pubmed/32466404
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom10060812
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