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Identification of 3,4-Dihydro-2H,6H-pyrimido[1,2-c][1,3]benzothiazin-6-imine Derivatives as Novel Selective Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase

Plasmodium falciparum’s resistance to available antimalarial drugs highlights the need for the development of novel drugs. Pyrimidine de novo biosynthesis is a validated drug target for the prevention and treatment of malaria infection. P. falciparum dihydroorotate dehydrogenase (PfDHODH) catalyzes...

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Bibliografske podrobnosti
izdano v:Int J Mol Sci
Main Authors: Hartuti, Endah Dwi, Sakura, Takaya, Tagod, Mohammed S. O., Yoshida, Eri, Wang, Xinying, Mochizuki, Kota, Acharjee, Rajib, Matsuo, Yuichi, Tokumasu, Fuyuki, Mori, Mihoko, Waluyo, Danang, Shiomi, Kazuro, Nozaki, Tomoyoshi, Hamano, Shinjiro, Shiba, Tomoo, Kita, Kiyoshi, Inaoka, Daniel Ken
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2021
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC8268581/
https://ncbi.nlm.nih.gov/pubmed/34281290
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms22137236
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