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A Box of Chemistry to Inhibit the MEN1 Tumor Suppressor Gene Promoting Leukemia

Targeting protein‐protein interactions (PPIs) with small‐molecule inhibitors has become a hotbed of modern drug development. In this review, we describe a new class of PPI inhibitors that block menin from binding to MLL proteins. Menin is encoded by the MEN1 tumor suppressor, but acts as an essentia...

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Pubblicato in:ChemMedChem
Autori principali: Ozyerli‐Goknar, Ezgi, Nizamuddin, Sheikh, Timmers, H. T. Marc
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8252030/
https://ncbi.nlm.nih.gov/pubmed/33534953
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.202000972
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