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Mechanistic Investigations of Metallo‐β‐lactamase Inhibitors: Strong Zinc Binding Is Not Required for Potent Enzyme Inhibition

Metallo‐β‐lactamases (MBLs) are zinc‐dependent bacterial enzymes that inactivate essentially all classes of β‐lactam antibiotics including last‐resort carbapenems. At present there are no clinically approved MBL inhibitors, and in order to develop such agents it is essential to understand their inhi...

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Détails bibliographiques
Publié dans:ChemMedChem
Auteurs principaux: Wade, Nicola, Tehrani, Kamaleddin H. M. E., Brüchle, Nora C., van Haren, Matthijs J., Mashayekhi, Vida, Martin, Nathaniel I.
Format: Artigo
Langue:Inglês
Publié: John Wiley and Sons Inc. 2021
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC8248298/
https://ncbi.nlm.nih.gov/pubmed/33534956
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.202100042
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