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A Pan-Inhibitor for Protein Arginine Methyltransferase Family Enzymes

Protein arginine methyltransferases (PRMTs) play important roles in transcription, splicing, DNA damage repair, RNA biology, and cellular metabolism. Thus, PRMTs have been attractive targets for various diseases. In this study, we reported the design and synthesis of a potent pan-inhibitor for PRMTs...

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Dettagli Bibliografici
Pubblicato in:Biomolecules
Autori principali: Iyamu, Iredia D., Al-Hamashi, Ayad A., Huang, Rong
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2021
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8230315/
https://ncbi.nlm.nih.gov/pubmed/34201091
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom11060854
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