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Force field optimization guided by small molecule crystal lattice data enables consistent sub-Angstrom protein-ligand docking

Accurate and rapid calculation of protein-small molecule interaction free energies is critical for computational drug discovery. Because of the large chemical space spanned by drug-like molecules, classical force fields contain thousands of parameters describing atom-pair distance and torsional pref...

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Detalhes bibliográficos
Publicado no:J Chem Theory Comput
Main Authors: Park, Hahnbeom, Zhou, Guangfeng, Baek, Minkyung, Baker, David, DiMaio, Frank
Formato: Artigo
Idioma:Inglês
Publicado em: 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8218654/
https://ncbi.nlm.nih.gov/pubmed/33577321
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.0c01184
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