Loading...

Synthesis of 2-oxoglutarate derivatives and their evaluation as cosubstrates and inhibitors of human aspartate/asparagine-β-hydroxylase

2-Oxoglutarate (2OG) is involved in biological processes including oxidations catalyzed by 2OG oxygenases for which it is a cosubstrate. Eukaryotic 2OG oxygenases have roles in collagen biosynthesis, lipid metabolism, DNA/RNA modification, transcriptional regulation, and the hypoxic response. Aspart...

Full description

Saved in:
Bibliographic Details
Published in:Chem Sci
Main Authors: Brewitz, Lennart, Nakashima, Yu, Schofield, Christopher J.
Format: Artigo
Language:Inglês
Published: The Royal Society of Chemistry 2020
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC8179049/
https://ncbi.nlm.nih.gov/pubmed/34163896
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc04301j
Tags: Add Tag
No Tags, Be the first to tag this record!