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SAR Insights Into TET2 Catalytic Domain Inhibition: Synthesis of 2-Hydroxy-4-Methylene-pentanedicarboxylates

The TET enzyme family of Ten-Eleven Translocation methylcytosine (5mC) dioxygenases comprising 3 members, TET1–3, play key roles in DNA demethylation. These processes regulate transcription programs that determine cell lineage, survival, proliferation, and differentiation. The impetus for our invest...

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Détails bibliographiques
Publié dans:Bioorg Med Chem
Auteurs principaux: Tiwari, Anand D., Guan, Yihong, Grabowski, Dale R., Maciejewski, Jaroslaw P., Jha, Babal K., Phillips, James G.
Format: Artigo
Langue:Inglês
Publié: 2021
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC8171112/
https://ncbi.nlm.nih.gov/pubmed/33894507
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2021.116141
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